Cell-permeable calmodulin (CaM) agonist that binds to the EF-hand/Ca2+-binding site; produces CaM-dependent activation of phosphodiesterase. Also binds to cytoplasmic sites on other Ca2+ channels, including NMDA and HIV-1 gp120-activated channels, inhibiting Ca2+-mediated cytotoxicity and apoptosis (IC50 = 52 μM). Shown to protect pancreatic acinar cells from gossypol induced necrosis. Inhibits VLA-5-mediated adhesion of mast cells to fibronectin in vitro and attenuates inflammatory cell influx in guinea pig lung in vivo.

二烯丙基三硫化物是大蒜中发现的一种有机多硫化物，可作为 H2S 供体。

TAK-700 (Orteronel) 是一种有效且高度选择性的人类 17, 20-裂解酶抑制剂，IC50 为 38 nM，其选择性比其他 CYP（例如 11-羟化酶和 CYP3A4）高 1000 倍。